G Protein-Coupled Receptors (GPCRs) Bioassay Services

G protein-coupled receptors (GPCRs) play important roles in cellular physiology and they are popular drug targets for various diseases. About 40% of approved drugs on the market belong to this category. Drug candidate screening and profiling is a critical step in GPCR-centered drug discovery. GenScript offers a comprehensive platform to speed up your GPCR drug discovery.

Key Features

  • Over 150 different GPCR functional cell lines
  • Customized GPCR stable cell line construction
  • Multiple assay formats including calcium flux, cAMP determination, and Luciferase reporter gene assays
  • Determine drug potency and efficacy in agonist, antagonist, inverse agonist and allosteric modulator modes
  • Stringent QC standards with competitive prices
  • Short turnaround time

Figure 1. GenScript offers multiple functional assays to characterize your samples for agonist, inverse agonist, antagonist and allosteric modulator activities.

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